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Cholesterol Absorption Inhibitors

Small intestine absorbs cholesterol from diet; Cholesterol absorption inhibitor medication reduces the cholesterol by inhibiting absorption of dietary cholesterol. Cholesterol absorption inhibitors can decrease LDL, slightly decrease triglycerides, and slightly increase HDL.

Cholesterol absorption inhibitor drug

  • Ezetimibe (Zetia).
  • Zetia can be useful in combination with any of the statin drugs.

Whom Zetia drug can benefit?

  • Not reaching their cholesterol targets on maximal doses of other medications,
  • If you are unable to tolerate other cholesterol, medication drugs because of liver, muscle, or other side effects.

How do you take Zetia drug?

  • Take this medication drug at the same time each day with or without food.
  • If you are taking Sequestrants, it should take at least two hours before or four hours after taking Zetia.

Possible side effects of Zetia drugs

  • The most common side effects related to the use of Zetia include stomach irritation, headache, abdominal pain, constipation, or diarrhea.
  • If taken along with a statin medication drug, the possible side effects may be headache, fatigue, abdominal pain, constipation, diarrhea, nausea, muscle weakness.

Stop the statin medication drug and contact the doctor immediately if experience: Muscle tenderness or soreness, unexplained muscle pain, general malaise, fatigue and weakness, and Fever.